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| 13-(苯并噻唑-2-基)-6,12-环亚胺二苯并[1,5]二氮杂环辛 衍生物的合成及杀菌活性 |
| Synthesis and Bactericidal Activity of 13-(benzothiazol-2-yl)-6H,12H-6,12-epiminodibenzo[1,5]diazocine derivatives |
| 投稿时间：2024-03-19 修订日期：2024-06-09 |
| DOI： |
| 中文关键词: 6,12-环亚胺二苯并[1,5]二氮杂环辛 2-氨基苯甲醛 2-氨基苯并噻唑 串联环化 杀菌活性 |
| 英文关键词: 6,12-epiminodibenzo[b,f][1,5]diazocine 2-aminobenzaldehyde 2-aminobenzothiazole cascade cyclization bactericidal activity |
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| 中文摘要: |
| 具有特殊三维结构的氮杂桥环化合物在医药、材料、超分子化学等领域有着广阔的应用前景和重要的研究意义。本文建立了以邻伯氨基苯甲醛和芳胺为原料构筑氮杂桥环的方法，合成了35个具有Y型空间结构的13-(苯并噻唑-2-基)-6,12-环亚胺二苯并[b,f][1,5]二氮杂环辛衍生物，并测试了它们对七种农作物细菌性病害的杀菌活性。该方法反应条件温和、原料易得，为开发结构新颖、具有杀菌活性的氮杂桥环化合物提供了新思路。 |
| 英文摘要: |
| Bridged cyclic compounds containing nitrogen atoms with special three-dimensional structures have broad application and important research significance in various fields such as medicine, materials, and supramolecular chemistry. In this paper, a method for constructing bridged cyclic compounds containing nitrogen atoms was established based on o-primaryaminobenzaldehyde and aromatic amine. Thirty-five 13-(benzothiazol-2-yl)-6H,12H-6,12-epiminodibenzo[b,f][1,5]diazocine derivatives with Y-shaped spatial structures were synthesized, and their bactericidal activity against seven crop bacterial diseases was tested. This approach has the advantages of mild reaction condition and easy availability of reactants. It provides new insight into the development of bridged cyclic compounds containing nitrogen atoms with novel structure and bactericidal activity. |
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